Basf Se Corporation

Boehringer Ingelheim Animal Health USA Inc.

Merial Limited

Karsten Körber

Wolfgang Von Deyn

Deborah L Culbertson

Florian Kaiser

Joachim Dickhaut

Nina Gertrud Bandur

Arun Narine

Prashant Deshmukh

Koshi Gunjima

Matthias Pohlman

Douglas D Anspaugh

Paul Allen Neese

Steffen Groβ

Ralph Paulini

Michael Rack

Michael Puhl

Egon Haden

Jochen Dietz

Henricus Maria Martinus Bastiaans

Hassan Oloumi-Sadeghi

Ronan Le Vezouet

Gemma Veitch

Markus Kordes

Maximilian Dochnahl

Timo Frassetto

Steffen Gross

Birgit Gockel

Franz-Josef Braun

Jean-Yves Wach

Christian Defieber

Jürgen Langewald

Joachim Schmidt-Leithoff

Delphine Breuninger

Franz Josef Braun

Sebastian Sörgel

Pascal Bindschädler

Martin John McLaughlin

Sarah Thompson

Cecille Ebuenga

Nancy B Rankl

Swetlana Derksen

Martin John Mclaughlin

Christian Rein

Michael David

W David Rogers

Steffen Groß

Daniel SÄLINGER

Kenichi Kojima

Martinjohn Mclaughlin

Paul Neese

The present invention relates to thiophene- or furan-substituted isothiazoline compounds of formula I wherein the variables are as defined in the claims and description. The compounds are useful for combating or controlling invertebrate pests, in particular arthropod pests and nematodes. The invention also relates to a method for controlling invertebrate pests by using these compounds and to plant propagation material and to an agricultural and a veterinary composition comprising said compounds.

Thiophene- or furan-substituted isothiazoline compounds as pesticides

The present invention relates to naphthyl- or isoquinolinyl-substituted isothiazoline compounds of formula I wherein the variables are as defined in the claims and description. The compounds are useful for combating or controlling invertebrate pests, in particular arthropod pests and nematodes. The invention also relates to a method for controlling invertebrate pests by using these compounds and to plant propagation material and to an agricultural and a veterinary composition comprising said compounds.

Naphthyl- or isoquinolinyl-substituted isothiazoline compounds

The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

N-acylimino heterocyclic compounds

The present invention relates to N-thioanthranilamide compounds of formula (I), and the stereoisomers, N-oxides and agriculturally or veterinarily acceptable salts thereof, wherein the substituents are as defined in the description. The present invention further relates to a method for combating or controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites, to a process for the preparation of a composition for treating infested or infected animals and/or for protecting animals against infestation or infection by parasites, and to a compound according to the invention for use as a medicament.

N-thio-anthranilamide compounds and their use as pesticides

The invention relates to N-substituted hetero-bicyclic compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to methods and uses of these N-substituted hetero-bicyclic compounds, and of compositions comprising thereof, for combating and controlling animal pests. Furthermore the invention relates also to pesticidal methods of applying such N-substituted hetero-bicyclic compounds. The N-substituted hetero-bicyclic compounds of the present invention are defined by the following formula I: wherein A, B, X, Het, R, R, W, W, Wand Ware defined as in the description.

N-substituted hetero-bicyclic compounds and derivatives for combating animal pests II

The invention relates to pyridylidene compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to methods and uses of these N-substituted pyridylidene compounds, and of compositions comprising thereof, for combating and controlling animal pests. Furthermore the invention relates also to pesticidal methods of applying such N-substituted pyridylidene compounds. The N-substituted pyridylidene compounds of the present invention are defined by the following formula I: wherein X, Het, R, R, R, Rand Rare defined as in the description.

N-substituted pyridinylidenes for combating animal pests

The present invention relates to substituted pyrazole-containing compounds of formula (I), and the stereoisomers and salts thereof, wherein the substituents are as defined in the description. The present invention further relates to a method for combating or controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites, to a process for the preparation of a composition for treating infested or infected animals and/or for protecting animals against infestation or infection by parasites, and to a compound according to the invention for use as a medicament.

Substituted pyrazole-containing compounds and their use as pesticides

The present invention relates to N-thio-anthranilamide compounds of the formula (I), the stereoisomers, the salts, the tautomers and the N-oxides thereof, wherein Ris halogen or halomethyl; Ris hydrogen, halogen or cyano; Ris hydrogen, C-Calkyl, C-Chaloalkyl, C-C-alkenyl or the like; Ris halogen; Rand Rindependently of each other are optionally substituted C-C-alkyl, C-C-cycloalkyl, C-C-alkenyl, C-C-alkynyl, phenyl, or together represent an (hetero)aliphatic chain, or the like; k is 0 or 1. The present invention further relates to a method for combating or controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites, to a process for the preparation of a composition for treating infested or infected animals and/or for protecting animals against infestation or infection by parasites, and to a compound according to the invention for use as a medicament.

The present invention relates to a process for preparing an N-substituted 1H-pyrazole-5-carbonylchloride compound of the formula (I) in which Ris hydrogen, halogen, cyano, C-C-alkyl, C-C-fluoroalkyl, C-C-cycloalkyl, C-C-fluorocycloalkyl, C-C-alkenyl, C-C-fluoroalkenyl, C-C-alkoxy, C-C-fluoroalkoxy, C-C-fluoroalkoxy-C-C-alkyl, phenyl and the like; each Ris independently selected from halogen, C-C-alkyl, C-C-fluoroalkyl, C-C-cycloalkyl, C-C-fluorocycloalkyl, C-C-alkenyl, C-C-fluoroalkenyl, C-C-alkoxy, phenyl and the like; r is 0, 1, 2, 3 or 4;comprising the steps of 

Process for preparing N-substituted 1H-pyrazole-5-carbonylchloride compounds

The present invention relates to a method for controlling invertebrate pests which method comprises treating the pests, their food supply, their habitat or their breeding ground or a plant, seed, soil, area, material or environment in which the pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from pest attack or infestation with a pesticidally effective amount of a pyrazole compound of formulae I or II or a salt or an N-oxide thereof, wherein A is a pyrazole radical of the formulae A1 or A2, wherein # denotes the binding; D is a 5- or 6-membered heterocyclic radical fused to the pyrazole moiety; R, Rand Rare H, halogen, CN, NO, C-C-alkyl, C-C-alkenyl, C-C-alkynyl, etc.; n is 0 to 4; or two radicals Rbound to the same ring-member may form an oxo substituent, or two radicals Rbound to adjacent ring-members may form a 3- to 7-membered fused cyclic radical; B is N or CR, wherein Ris H, halogen, CN, NO, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, etc.; Xis S, O or NR, wherein Ris H, C-C-alkyl, etc.; Xis O, NRRor S(O)R, wherein m is 0, 1 or 2; Ris C-C-alkyl, C-C-haloalkyl, C-C-cycloalkyl, etc.; R, Rare H, C-C-alkyl, C-C-haloalkyl, C-C-cycloalkyl, etc.; Ris C-C-alkyl, C-C-haloalkyl, C-C-cycloalkyl, etc.; Ris H, CN, C-C-alkyl, C-C-haloalkyl, C-C-cycloalkyl, etc.; R, Rand Rare H, halogen, CN, NO, C-C-alkyl, C-C-haloalkyl, C-C-alkoxy, etc., to a method for protecting plant propagation material and/or the plants which grow threfrom, to plant propagation material comprising at least one compound of formulae I or II, to a method for treating or protecting an animal from infestation or infection by parasites, to novel pyrazole compounds of formulae I or II and agricultural composition containing those compounds. 

Pyrazole compounds for controlling invertebrate pests

The present invention relates to the 3-arylquinazolin-4-one compounds of the formula I and the salts thereof, wherein The invention also relates to the use of novel compounds of formula I for combating invertebrate pests and to a method for controlling invertebrate pests. The invention also relates to a plant propagation material and to an agricultural composition comprising a 3-arylquinazolin-4-one compound of formula I.

3-arylquinazolin-4-one compounds for combating invertebrate pests

The present invention relates to pyrazole compounds of formulae I or II and the salts and N-oxides thereof, wherein A is a pyrazole radical of formulae A1, A2 or A3, wherein # denotes the binding site; R, R, R, Rare H, halogen, CN, NO, C-C-alkyl and the like; R, Rare H, halogen, CN, NO, C-C-alkyl, and the like; R, R, Rare H, CN, NO, C-C-alkyl, and the like; T is C(R) or N; U is C(R) or N; V is C(R) or N; W is C(R) or N; with the proviso that at least one of the groups T, U, V and W is N; R, R, R, Rare H, halogen, C-C-alkyl and the like; Xis S, O or NR, wherein Ris selected H, C-C-alkyl and the like; Xis OR, NRR, S(O)R, wherein m is 0, 1 or 2, Ris C-C-alkyl, C-C-haloalkyl and the like, R, Rare H, C-C-alkyl, C-C-haloalkyl and the like, or Rand Rtogether with the nitrogen atom to which they are bound form a heterocycle, and Ris C-C-alkyl, C-C-haloalkyl, C-C-cycloalkyl and the like; and Ris H, CN, C-C-alkyl and the like.The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plan propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

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Eppelheim, Germany

Karsten Körber