Novartis Animal Health Us, Inc.

Novartis Ag

Navartis Animal Health Us, Inc.

Jacques Bouvier

Pierre Ducray

Thomas Goebel

Tania Cavaliero

Catherine Christinaz

Olivier Froelich

Steve Nanchen

Nicola Di Criscio

Corinne Durano

Noëlle Gauvry

Sandra Schorderet Weber

François Pautrat

Maurizio Schwarzenbach

Jorg Fruchtel

Matthias Keller

Catherine Kolly

Urs M&uuml;ller

Corina Bergamin

Richard Hunter

John Marshall

Maike Lohrmann

Beatrice Bapst

Jörg Früchtel

Maike Renner

Jean-Luc Perret

Martin Fink

John Gerard Mchenery

The present invention is directed to a non-therapeutical process for deterring vermin, which is based on the usage of the largely known beta amino-alcohol derivatives of formula (I) as described herein. Further, the present invention is directed to corresponding vermin-deterring compositions which contain these substances as the active ingredient, compounds of the formula (I) for the preparation of vermin-deterring compositions, and the use of compounds of formula (I) in the defense against vermin.

Composition for repelling and deterring vermin

The invention relates to new pyrimidine compounds of formula (1) wherein the variables have the meaning as indicated in the claims; in free form and in salt form; and optionally the enantiomers and geometrical isomers thereof. The compounds of formula (1) are useful in the control of parasites, in particular ectoparasites, in and on warmblooded animals. 

Pyrimidine derivatives and their use as pesticides

The invention describes essentially a non-therapeutical process for deterring vermin, which is based on the usage of the largely known beta amino-alcohol derivatives of formula (I), as defined herein before. Furthermore, it describes the corresponding vermin-deterring compositions which contain these substances as the active ingredient, compounds of the formula (I) for the preparation of vermin-deterring compositions, and the use of compounds of formula (I) in the defense against vermin. Thus, the invention describes how and in which form the compounds of the formula (I) or their acid addition salts are used to deter vermin from materials, places or warm-blooded animals. 

The present invention relates to the use of compounds of formula (I), wherein R, X, Y, Z and m are as defined in the description, in the free form or in salt form either alone or in combination with a vaccine component, for controlling fish parasites, in particular sea lice. 

Use of oxazole derivatives for controlling fish parasites

Compounds of formula (I) are described for deterring vermin, wherein R is unbranched or branched C-Calkyl, which is unsubstituted or substituted by halogen, cyano or nitro; R1 and R2 are unbranched or branched C-Calkyl, preferably C-Calkyl, which is unsubstituted or substituted by halogen, cyano or nitro; and X and Y, independently of one another, are a straightchain or branched alkylene bridge with 1 to 20 carbon atoms, preferably an alkylene bridge with 1 to 3 carbon atoms, which is unsubstituted or substituted by halogen, cyano or nitro. Furthermore, an essentially non-therapeutical process for deterring vermin is described, which is based on the usage of these compounds, as well as verminrepellent compositions containing these compounds as the active ingredient, and finally the use of these compounds for producing vermin-deterring compositions and their usage in deterring vermin from animals, humans and objects. New compounds within the scope of formula (I) are also described. 

Vermin-repellant compositions and compounds

The invention relates to compounds of the general formula and optionally the enantiomers thereof. These compounds have advantageous pesticidal properties. They are especially suitable for controlling parasites in warm-blooded animals.

Benzamidoacetonitriles and their use as antiparasitics

The invention relates to the use of aminoacetonitrile compounds of formula (I), wherein R, R, R, R, R, R, A, m and n have the significances given in claim, in the control of endoparasites, especially helminths, in warm-blooded productie livestock and domestic animals.

Organic compounds

The invention relates to compounds of the general formula in which R, R, R, R, R, W, X, A, A, a, b and c are as defined in the specification, and to any enantiomers thereof. The active ingredients have advantageous pesticidal properties. They are particularly suitable for controlling parasites in warm-blooded animals.

N-acylaminoacetonitrile derivatives and their use for controlling parasites

The invention relates to compounds of the general formula: (I) and optionally the enantiomers thereof. The active ingredients have advantages pesticidal properties. They are especially suitable for controlling parasites on warm-blooded animals.

Amidoacetonitrile compounds and their use as pesticides

The invention relates to compounds of the general formula (I), in which Ar, R, R, R, R, R, R, R, R, W, a, b and n are as defined in claim, and to any enantiomers thereof. The active ingredients have advantageous pesticidal properties. They are particularly suitable for controlling parasites in warm-blooded animals 

Amidoacetonitrile derivatives

The invention relates to compounds of formula I wherein R, R, R, R, R, R, R, R, R, W, X, A, A, a, b and c have the significances given in the specification, and optionally the enantiomers thereof. The active ingredients have advantageous pesticidal properties. They are especially suitable for controlling parasites on warm-blooded animals.

Amidoacetonitrile compounds

The invention relates to a composition for controlling a pest, including endoparasites, and more specifically helminths, of formula (I) in animals, and methods related to thereof.

Pharmaceutical composition containing aminocetonitrile compounds and the use thereof for the preparation of a pharmaceutical composition for the treatment of endoparasitic pests in animals

Pharmaceutical composition containing aminoacetonitril compounds and the use thereof for the preparation of a pharmaceutical composition for the treatment of endoparasitic pests in animals

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Neuchatel, Switzerland

Jacques Bouvier