Glaxosmithkline Intellectual Property (no.2) Limited

Anacor Pharmaceuticals, Inc.

Glaxo Group Limited

Ilaria Giordano

Jacob J Plattner

Vincent S Hernandez

Xianfeng Li

David Barros-Aguirre

Neil David Pearson

Alan Joseph Hennessy

Michael Richard Kevin Alley

David Thomas Davies

Carlos Alemparte-Gallardo

Gerald Brooks

Michael Richard Kevin (Dickon) Alley

Graham Elgin Jones

Steven Dabbs

Timothy James Miles

Israil Pendrak

Julia Castro Pichel

Robert A Daines

Jose Maria Fiandor Roman

Lihua(lily) Zhang

David Barros

James B Hoffman

Jason Anthony Rossi

Modesto J Remuiñan Blanco

Lluis Ballell

David Evan Davies

Substituted benzoxaboroles whose structure comprises Formula (III), wherein Ris selected from &#x2014;CH, &#x2014;CIICII, &#x2014;CII&#x2550;CII, &#x2014;CIICIICII, &#x2014;CH(CH), &#x2014;CHCH&#x2550;CH, and cyclopropyl, Rand Rare each independently selected from H, &#x2014;CH, &#x2014;CHCH, &#x2014;CHCHCH, and &#x2014;CH(CH); compositions containing such compounds, their use in therapy, including their use as anti-mycobacterial agents, for example in the treatment of a mycobacterial infection in a mammal, and methods for the preparation of such compounds, are provided.

4-substituted benzoxaborole compounds and uses thereof

Compounds of Formula II, wherein X is selected from chloro, fluoro, bromo and iodo, Rand Rare each independently selected from H, &#x2014;CH, &#x2014;CHCH, &#x2014;CHCHCH, or &#x2014;CH(CH); compositions containing them, their use in therapy, including their use as anti-mycobacterial agents, for example in the treatment of a mycobacterial infection in a mammal, and methods for the preparation of such compounds, are provided.

Tricyclic benzoxaborole compounds and uses thereof

Substituted benzoxaboroles whose structure comprises Formula (III), wherein Ris selected from &#x2014;CH, &#x2014;CHCH, &#x2014;CH&#x2550;CH, &#x2014;CHCHCH, &#x2014;CH(CH), &#x2014;CHCH&#x2550;CH, and cyclopropyl, Rand Rare each independently selected from H, &#x2014;CH, &#x2014;CHCH, &#x2014;CHCHCH, and &#x2014;CH(CH); compositions containing such compounds, their use in therapy, including their use as anti-mycobacterial agents, for example in the treatment of a mycobacterial infection in a mammal, and methods for the preparation of such compounds, are provided. 

Tricyclic nitrogen containing compounds and their use as antibacterials. Zand Zare independently selected from CH and N. 

Tricyclic nitrogen containing compounds as antibacterial agents

Bicyclic nitrogen containing compounds and their use as antibacterials.

Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones

Tricyclic nitrogen containing compounds of formula (I) and their use as antibacterials.

Tryclic nitrogen containing compounds and their use as antibacterials

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Hertfordshire, United Kingdom

Ilaria Giordano