Merial Limited

Boehringer Ingelheim Animal Health USA Inc.

Aventis Agriculture Limited

Boehringer Ingelheim Vetmedica Gmbh

Boehringer Ingelheim Pharma Gmbh & Co Kg

Aventis Agiziculture

Hyoung Ik Lee

Loic Patrick Le Hir De Fallois

Charles Q Meng

Alan Long

Douglas Edward Wilkinson

Greg Pacofsky

Philip Reid Timmons

Brent Christopher Beck

Robert Toms Jacobs

Scot Kevin Huber

Loïc Patrick Le Hir De Fallois

William Glenn Cawthorne, Jr

Mark Soll

Mark David Soll

Cyprian Okwara Ogbu

Adalberto A Perez De Leon

Adalberto Perez De Leon

Jean Robert Labrosse

Xinxi Zhan

Michel Mulhauser

Hannes Fiepko Koolman

Gregory Pacofsky

Cyprian O Ogbu

Loic Le Hir De Fallois

Jean-Robert Labrosse

Loic Le De Fallois

William Glenn Cawthorne

Loiec Patrick Le Hir De Fallois

The present invention provides cyclic depsipeptide compounds of formula (I) and compositions comprising the compounds that are effective against parasites that harm animals. The compounds and compositions may be used for combating parasites in or on mammals and birds. The invention also provides for an improved method for eradicating, controlling and preventing parasite infestation in birds and mammals.

Anthelmintic depsipeptide compounds

Cyclic depsipeptide compounds of formula (I) and compositions comprising the compounds are provided that are effective against parasites that harm animals, including humans. The compounds and compositions may be used for combating parasites in or on animals including mammals and birds. Also provided are improved methods for eradicating, controlling and preventing parasite infestation in animals, including birds and mammals.

The compound of formula I: compositions thereof, processes for their preparation, and their uses as pesticides.

Indazolylcyanoethylamino compound, compositions of same, method of making, and methods of using thereof

The present invention relates to pesticidal and parasiticidal isoxazoline of formula (I) and salts thereof: wherein variables R, P, Y and Q are described herein are as defined in the description. The invention also relates to parasiticidal and pesticidal compositions comprising the isoxazoline compounds of formula (I), processes for their preparation and their uses to prevent or treat parasitic infections or infestations in animals and as pesticides.

Pesticidal and parasiticidal pyrazole-isoxazoline compounds

This invention provides for compounds of the formula: wherein the variables are defined herein, or a stereoisomer, tautomer, N-oxide, hydrate, solvate, or salt thereof, compositions comprising these compounds, and method for the treatment, control or prevention of a parasitic infestation or infection in an animal in need thereof by administering an effective amount of these compounds to said animal.

Anthelmintic aza-benzothiophene and aza-benzofuran compounds

The present invention provides cyclic depsipeptide compounds of formula (I) wherein the stereochemical configuration of at least one carbon atom bearing the groups Cy, Cy, R, R, R, R, Rand Ris inverted compared with the naturally occurring cyclic depsipeptide PF1022A. The invention also provides compositions comprising the compounds that are effective against parasites that harm animals. The compounds and compositions may be used for combating parasites in or on mammals and birds. The invention also provides for an improved method for eradicating, controlling and preventing parasite infestation in birds and mammals.

The present invention provides cyclic depsipeptide compounds of formula (I) and compositions comprising the compounds that are effective against parasites that harm animals, including humans. The compounds and compositions may be used for combating parasites in or on animals including mammals and birds. The invention also provides for an improved method for eradicating, controlling and preventing parasite infestation in animals, including birds and mammals.

The present invention relates to novel dihydroazole of formula (I) and salts thereof: Wherein R, A, A, G, X and Y are as defined in the description, compositions thereof, processes for their preparation and their uses to prevent or treat parasitic infections or infestations in animals and as pesticides.

Antiparisitic dihydroazole compounds and compositions comprising same

Provided are 1-aryl-5-alkyl pyrazole compounds, of formula (I): wherein: Ris hydrogen, cyano, halogen, R, formyl, &#x2014;C(O)R, &#x2014;C(O)OR, &#x2014;C(O)NRR, or &#x2014;C(S)NH; Ris Ror &#x2014;S(O)R; Ris methyl, ethyl or C-Chaloalkyl; R, Rand Rare independently hydrogen, halogen, alkyl, haloalkyl, cyano or nitro; Ris halogen, alkyl, haloalkyl, alkoxy, haloalkyloxy, cyano, nitro, &#x2014;C(O)R, &#x2014;S(O)Ror SF; Z is a nitrogen atom or C&#x2014;R; Ris alkyl, haloalkyl, cycloalkyl or halocycloalkyl; Ris hydrogen, alkyl, haloalkyl or alkoxy; Ris hydrogen, alkyl, haloalkyl or alkoxy; Ris alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl or cycloalkyl; Ris alkyl or haloalkyl; Ris hydrogen, halogen, cyano, nitro, alkyl, haloalkyl, alkoxy or haloalkoxy; m is 0, 1 or 2; and n is 0, 1 or 2; or a salt thereof, the method of making compounds of formula (I) and the use of these compounds against ectoparasites, endoparasites and pests.

1-aryl-5-alkyl pyrazole derivative compounds, processes of making and methods of using thereof

Provided are improved processes for the preparation of 1-aryl pyrazole compounds of formula (I) and (IB): which are substituted at the 5-position of the pyrazole ring with a carbon-linked functional group. The process described are efficient and scalable and do not utilize hazardous sulfenyl halide reagents.

Processes for the preparation of 1-aryl-5-alkyl pyrazole compounds

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Cary, NC, United States of America

Hyoung Ik Lee