Hoechst Aktiengesellschaft

Hoechst Aktiengeselleschaft

Hermann J Gerhards

Bernward Scholkens

Adalbert Wagner

Rainer Henning

Klaus-Dieter Kampe

Herbert Siegel

Patricia Usinger

Heinz-Werner Kleemann

Wolfgang Raether

Burkhard Sachse

Holger Heitsch

Rudolf Lattrell

Walter Dittmar

Jean-Paul Vevert

Hans-Georg Alpermann

Ulrich Schacht

Margret Leven

Jochen Knolle

Rolf Geiger

Gerhard Breipohl

Reinhard Becker

Stephan Henke

Hansjorg Kruse

Hans G Alpermann

Jean-Claude Caille

Manfred Forsch

Klaus Wirth

Heinrich Christian Englert

Wilhelm Bartmann

Ulrich Lerch

Walter Durckheimer

Hans-Wolfram Fehlhaber

Wolfgang Linz

Elmar Schrinner

Rudolf Kunstmann

Hiristo Anagnostopulos

Franz Hock

Alfons Soder

Wolfgang Schaub

Fritz Bauer

Jens Stechl

Herbert Hartung

Peter Klatt

John-Claude Caille

Bernward Sch Olkens

Alfred Kreutzberger

Peptides having bradykinin antagonist action

A compound of the formula ##STR1## in which the symbols have the following meaning: X is a monocyclic radical having 3, 4 or 5 ring atoms,

Benzimidazole derivatives as angiotensin II receptor antagonists,

Imidazole derivatives with a biphenylsulfonylurea or biphenylsulfonylurethane side chain, process for their preparation and their use Compounds of the formula (I) ##STR1## in which R.sup.1 is, for example, ethyl,

Imidazole derivatives with a biphenylsulfonylurea or

Bradykinin peptides with modifications at the N terminus

Azole derivatives, process for their preparation, and their use Azole derivatives of the formula (I) ##STR1## in which A, L, O, R.sup.1, X, Y, Z and q have the meanings given, process for their preparation, pharmaceutical preparations and the use of the compounds are described. Azole derivatives of the formula I where the symbols have for example the following meanings:

Azole derivatives, process for their preparation and their use

Imidazo-fused iso- and heterocycles, process for their preparation, compositions containing them and their use A compound of the formula ##STR1## in which the symbols have the following meaning: X is a monocyclic radical having 3,4 or 5 ring atoms,

Imidazopyridine derivatives as angiotensin II receptor antagonists,

The invention relates to compounds of the formula ##STR1## in which X, Y and Z are identical or different and are N or CR.sup.2, L is an alkylene radical, q is 0 or 1, and A is the radical of a fused heterobicyclic compound. The invention furthermore relates to a process for preparing the said compounds, agents containing these, and the use thereof for angiotensin II receptors.

Substituted imidazoles

The invention relates to compounds of the formula I ##STR1## in which X, Y and Z are identical or different and are N or CR.sup.2, R.sup.1 and R.sup.2 are as defined in the description, L is an alkylene radical, q is 0 or 1, and A is the radical of a fused heterobicyclic compound. The invention furthermore relates to a process for preparing the said compounds, agents containing these, and the use thereof in the treatment of high blood pressure.

Substituted imidazoles, pharmaceutical compositions containing these,

The invention relates to compounds of the formula (I) ##STR1## in which X, Y and Z are identical or different and are N or CR.sup.2, and the other radicals have the meaning defined in the description, a process for the preparation thereof, agents containing these, and the use thereof.

Substituted azoles, a process for their preparation, and their use

Arylmethylazoles of the formula I ##STR1## in which Aryl is (substituted) phenyl or naphthyl;

Arylmethylazoles and their salts, agents which contain these compounds,

Arylmethylazole preparation processes

1-(1-Aryl-2-hydroxyethyl)-imidazoles and salts thereof, processes for the preparation thereof, medicaments containing these compounds, and the use thereof. The invention relates to 1-(1-aryl-2-hydroxyethyl)-imidazoles of the formula I ##STR1## in which R.sup.1, R.sup.2, R.sup.3, Q, W, X and Y have the meanings specified, and also to medicaments based on these compounds, in particular those having an antimycotic and an antidepressive action.

1-(1-aryl-2-hydroxyethyl)-imidazoles and salts thereof, medicaments

Arylmethylazoles and their salts, processes for their preparation,

2,4,6-Tris-tertiary-butylamino-1,3,5-triazine of the formula I ##STR1## for the prophylaxis and treatment of epilepsy and anxiety states, and the use for the preparation of a medicament for the prophylaxis and treatment of epilepsy and anxiety states, are described.

2,4,6-tris-tertiary-butylamino-1,3,5-triazine useful for the prophylaxis

New substituted phenylpiperazine derivatives of the formula I ##STR1## in which R.sup.1 and R.sup.2 have the indicated meaning, and their physiologically tolerated salts and a process for their preparation are described. The compounds exhibit sedative and aggression-inhibiting effects on livestock. Furthermore, compounds of the formula I' ##STR2## in which n, A, R.sup.2, R.sup.3 and R.sup.4 have the indicated meanings, and their physiologically tolerated salts are claimed for the sedation and inhibition of aggression of livestock.

Phenylpiperazine propyloxyquinolinones and methods for sedating and

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Hofheim am Taunus, Germany

Hermann J Gerhards