Eli Lilly and Company

Harold M Taylor

Kenneth S Hirsch

Charles David Jones

Robert G Suhr

Mark Alan Winter

This invention provides a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals by administering certain amine derivatives.

Method of inhibiting aromatase

This invention provides a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals by administering certain amine derivatives. Pharmaceutical formulations of the compounds are also provided.

This invention provides a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals which comprises administering certain imidazole derivatives.

This invention provides a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals by administering certain pyrazine derivatives. Pharmaceutical formulations of the pyrazine derivatives are also provided.

This invention provides a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals by administering certain pyridine derivatives.

This invention provides a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals by administering certain azole derivatives.

This invention provides a method of inhibiting aromatase and treating estrogen-dependent diseases in mammals by administering certain azole derivatives. Certain azole derivatives and their pharmaceutical formulations are also provided.

Aromatase inhibitors

This invention provides certain imidazole derivatives, their pharmaceutical formulations, and their use in a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals.

Aromatase inhibiting .alpha.,.alpha.-diphenyl-4(5)imidazole-methanes or

This invention provides certain azole derivatives and their pharmaceutical formulations. Also provided is a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals by administering the azole derivatives.

Aromatase inhibiting imidazole derivatives

This invention provides certain azole derivatives, their pharmaceutical formulations, and a method of inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals.

Aromatase inhibiting derivatives of

This invention provides certain isoxazole and isothiazole derivatives, their pharmaceutical formulations, and their use in inhibiting aromatase and treating or preventing estrogen-dependent diseases in mammals.

Isoxazolyl and isothiazolyl aromatase inhibitors

A method of reducing the vigor of aquatic weeds and algae makes use of a class of 3-phenyl-4(1H)-pyridones and pyridinethiones. The new compounds are characterized by a methyl group on the nitrogen, and usually bear a 5-substituent chosen from a class which is described herein. The phenyl ring may be substituted. The compounds effectively control aquatic weeds and algae, and kill the plants slowly, so that their decomposition does not deplete oxygen in the treated body of water.

Method of controlling aquatic weeds and algae

A class of 1-alkyl-3-phenylpyridinium salts are useful herbicides. The compounds bear a meta-substituent on the phenyl ring and optional 4- and 5-substituents.

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Indianapolis, IN, United States of America

Harold M Taylor