Sandoz Gmbh

Sandoz Ltd., (sandoz Ag)

Novartis Corporation

Fritz Schaub

Hans-Peter Schelling

Martin Eberle

Gerald Wayne Craig

Rupert Schneider

Hanspeter Schelling

Clemens Lamberth

This invention relates to novel 2-(4-pyrazolyloxy-pyrimidin-5-yl) acetic acid derivatives of formula I ##STR1## wherein R.sub.1 is hydrogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, C.sub.1-4 alkylthio, C.sub.3-6 cycloalkyl, or di-C.sub.1-4 alkylamino,

2-(4-pyrazolyloxy-pyrimidin-5-yl) acetic acid derivatives

This invention relates to compounds of formula I ##STR1## wherein R.sup.1 is C.sub.1-4 alkoxy or --NR.sup.8 R.sup.9 ;

.alpha.-pyrimidinyl acrylic acid derivatives

This invention relates to 2-(4-alkylthio-pyrimidin-5-yl)-acetic acid derivatives; fungicidal compositions comprising such compounds and a method of combating phytopathogenic fungi comprising applying such compounds to the fungi or their habitat.

4-alkylthio-pyrimidin-5-ylacetic acid derivates

The invention discloses compounds of formula I ##STR1## the use of such compounds for the control of phytopathogens, composition for facilitating such use, and the preparation of the compounds of formula I.

The invention discloses compounds of formula I It has now been found that compounds of formula I ##STR1## wherein R.sub.1 is hydrogen, methyl, ethyl or trifluoromethyl, and

Pyrimidinyl acrylic acid derivatives

The invention compounds of formula I ##STR1## wherein R is H, C.sub.1-4 alkyl; optionally substituted aryl or CF.sub.3 ;

Pyrazoles, fungicidal compositions and use

The invention provides novel .alpha.-aryl- or -aralkyl-.alpha.-(cycloalkyl-alkyl)-1H-azole-1-ethanols, in which the alkyl moiety linking the cycloalkyl group to the ethanol group is substituted or branched at the carbon atom adjacent to the C(OH) group, which are useful as plant fungicides and for treating fungus diseases in man and animals. Other objects of the invention are plant fungicidal, pharmaceutical and veterinary compositions comprising such novel compounds and methods of combatting phytopathogenic fungi or fungus diseases with the aid of said novel compounds.

.alpha.-phenyl-.alpha.-cyclopropylalkyene-1H-imidazole- and 1,2,4

.alpha.-phenyl- or benzyl-.alpha.-cyclopropylalkylene-1H-imidazole- and

The invention provides novel .alpha.-(ethynyl substituted phenyl)-.alpha.-hydrocarbyl-1H-azole-ethanols wherein the azole group is 1,2,4-triazol-1-yl or imidazol-1-yl, the ethynyl group is unsubstituted or substituted and the phenyl group may bear an additional substituent and ethers thereof, which are useful as fungicides.

Fungicidal .alpha.-(alkynylphenyl)azole ethanol compounds

Benzodioxan derivatives of formula, ##STR1## in which R is a group of formula A ##STR2## or of formula B,

Ether substituted benzodioxan derivatives

The present invention concerns novel aromatic long chain alkyl ethers and thioethers of the formula, ##STR1## wherein R.sub.1 is a hydrocarbon group,

Polyether substituted 3,4-methylenedioxybenzenes

The present invention concerns novel aromatic long chain alkenyl ethers and thioethers of the formula: ##EQU1## wherein R.sub.1 is a hydrocarbon group,

Ether and thioether substituted 3,4-alkylenedioxybenzenes

The present invention concerns novel compounds of the formula: ##EQU1## wherein R.sub.1 to R.sub.9 have various significances including e.g. alkyl, X and Y include O and S and s, v, w and z are O or whole numbers and Ar.sub.1 is a formyl phenyl radical. The compounds possess insecticidal properties.

Ether of thioether substituted benzaldehydes

The present invention concerns the use of the compounds of the formula: ##EQU1## wherein R.sub.1 to R.sub.9 have various significances including e.g. alkyl, X and Y include O and S, and s, v, w and z are O or whole numbers and Ar.sub.1 is substituted phenyl, as insecticides, and insecticidal compositions containing said compounds as active agent.

Composition and method for combating insects with alkylenedioxyphenyl

The present invention concerns unsaturated ethers or thioethers of the formula: ##EQU1## wherein R.sub.1 is an aliphatic or alicyclic hydrocarbon, R.sub.2 and R.sub.3 are H or alkyl, Y is cyano, amido, a ketone or an acid ester, ##EQU2## is an ether, thioether or a saturated or unsaturated c--c bond and n is an integer, which exhibit insecticidal properties.

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Aesch, Switzerland

Fritz Schaub