Syngenta Crop Protection, Inc.

Merial Limited

Syngenta Corporation

Syngenta Corp Protection LLC

Fiona Murphy Kessabi

Laura Quaranta

Thomas Pitterna

Pierre Marcel Jung

Ottmar Franz Hueter

Peter Maienfisch

Jerome Yves Cassayre

Hans-Georg Brunner

Renaud Beaudegnies

Fredrik Cederbaum

Hans Tobler

Roger Salmon

Jérôme Yves Cassayre

Ewan James Turner Chrystal

Patrick J Crowley

David Philip Bacon

Olivia Anabelle Sageot

David William Langton

Gordon Richard Munns

Jayant Umarye

Andrew Jonathan Knee

Pierre Jung

Jérôme Cassayre

Compounds of the general formula (I), wherein the substituents are as defined in claim, are useful as fungicides. 

Saturated and insaturated bi- or tricyclic aryloxyacetamine derivatives and their use as fungicides

Fungicidal compounds of the general formula (I), wherein the substituents are as defined in claim. 

Fungicides

Compounds of the general Formula (1) wherein the substituents are as defined in claim, are useful as fungicides. 

Quinoline derivatives and their use as fungicides

What is described are a compound of the formula wherein

Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4&#x2033;-or 4'-position

Compounds of the formula wherein the substituents are as defined in the claims, are useful as fungicides. 

I-alkynyl 2-aryloxyalkylamides and their use as fungicides

Compounds of the general formula (I); wherein the substituents are as defined in claim, are useful as fungicides. 

Acetamide compounds as fungicides

Certain derivatives of avermectin, avermectin monosaccharide and avermectin aglycone, having on the 4&#x2033;, 4' or 13 position, respectively, a 6-membered cyclic acetal with a substituent on position 2, that are useful in controlling pests, in particular pests that are harmful to crop plants and to its propagation material, such as representatives of the class insecta, the order acarina and the class nematode, are provided. 

Derivatives of avermectin, avermectin monosaccharide and avermectin aglycone

Avermectin B1 and avermectin B1 monosaccharide derivative compounds having an alkoxymethyl substituent in the 4&#x2033;- or 4'-position; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions are provided.

Avermectin B1 and avermectin B1 monosaccharide derivatives having an alkoxymethyl substituent in the 4&#x2033; -or 4'-position

Described is a compound of the formula (I) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R, is C-Calkyl, C-Ccycloalkyl or C-Calkenyl; and either (A) Ris &#x2014;N(R)R, and (1) X is 0, wherein Ris, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C-Calkyl, and Ris, for instance, mono- to pentasubstituted C-Calkyl, unsubstituted or mono- to pentasubstituted C-Ccycloalkyl; or (2) X is S, wherein Ris, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C-Calkyl, and Ris, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C-Calkyl; or (3) X is 0 or S, wherein Rand Rtogether are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) Ris OR, X is 0 or S, wherein Ris, for instance, C-Calkyl, mono- to pentasubstituted C-Calkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity. 

Avermectins and avermectin monosacharides substituted in the 4'-and 4&#x2033; position having pesticidal properties

Avermectin and avermectin monosaccharaide compounds, derivatives, and compositions thereof are provided as well as processes for preparing such compounds, derivatives, and compositions. Intermediates in the preparation of avermectin and avermectin monosaccharaide derivatives and methods of controlling pests are also provided. The avermectin and avermectin monosaccharaide derivatives are demonstrated as useful in controlling pests, in particular pests that are harmful to crop plants and to its propagation materials, such as representatives of the class insecta, the order Acarina and the class nematede.

Avermectin and avermectin monosaccharide substituted in the 4&#x2033;- and 4&#x2033; position respectively

What is described are a compound of the formula (I) Wherein U is &#x2014;N(R)ORor &#x2014;N(O)&#x2550;C(R)R); n is 0 or 1; X&#x2014;Y is &#x2014;CH&#x2550;CH&#x2014; or &#x2014;CH&#x2014;CH&#x2014;; Ris C-Calkyl, C-Ccycloalkyl or C-Calkenyl; Rand Rare, for example; independently from each other, &#x2014;Q, &#x2014;C(&#x2550;O)&#x2014;Z&#x2014;Q or &#x2014;CN; Rand Rare, independently from each other, &#x2014;Q, &#x2014;C(&#x2550;O)&#x2014;Z&#x2014;Q or &#x2014;CN; or Rand Rtogether are a three- to seven membered alkylene or alkenylene bridge, which is unsubstituted or mono- to tri-substituted; Z is a bond, O or &#x2014;NR&#x2014;; Q is H, C-Calkyl, C-Calkenyl, C-Calkynyl, C-C-Cycloalkyl, C-C-cycloalkenyl, aryl, or heterocyclyl, which are unsubstituted or mono- to pentasubstituted; Ris for example H, C-Calkyl, hydroxy-C-Calkyl, C-Ccycloalkyl or C-Calkenyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions. 

Avermectin and avermectin monosaccharide derivatives substituted in the 4&#x2033;-or 4'-position having pesticidal properties

Disclosed are compounds of the formulain which n is 0 or 1; X&#x2014;Y is &#x2014;CH&#x2550;CH&#x2014; or &#x2014;CH&#x2014;CH&#x2014;; Z is &#x2014;C(&#x2550;O)&#x2014;, &#x2014;C(&#x2550;S)&#x2014; or &#x2014;SO&#x2014;; Ris C-Calkyl, C-Ccycloalkyl or C-Calkenyl; and Ris R-Z-, R&#x2014;O-Z-, Ror -Z-N(R)(R); Q is O or &#x2014;N&#x2014;R; Rand Rare for example H, CCalkyl, C-Calkenyl, C-Calkynyl, C-Czcycloalkyl, C-Ccycloalkenyl, aryl or heterocyclyl; Ris for example H, C-Calkyl, hydroxy-C-Calkyl, C-Ccycloalkyl, C-Calkenyl, C-Calkynyl, phenyl or benzyl; Rand Rare for example, H, unsubstituted or mono- to pentasubstituted C-Calkyl, unsubstituted or mono- to pentasubstituted C-Calkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides. 

Avermectin and avemectin monosaccharide derivatives substituted in the 4&#x2033;-  or 4'-position having pesticidal properties

A compound of formula (I); that has the S-configuration at the 4&#x2033;-position and wherein the bond between carbon atoms 22 and 23 is a single or a double bond; Ris C-Calkyl, C-Ccycloalkyl; or C-Calkenyl; Ris H, or, for example, unsubstituted or mono- to penta-substituted C-Calkyl, C-Calkenyl, C-Calkynyl or C-Calkoxy-C-Calkyl; Ris H or, for example, C-Calkyl; X is a bond, O, NRor S; and Z is C&#x2550;O, C&#x2550;S or S0; and, where applicable, E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for the preparation of and the use of those compounds and their isomers and tautomers; starting materials for the preparation of the compounds of formula (I); pesticidal compositions in which the active ingredient has been selected from those compounds and their tautomers; and a method of controlling pests using those compositions are described. 

4&#x2033;-deoxy-4&#x2033;-(S)-amido avermectin derivatives

A compound of formula (I) wherein the bond between carbon atoms 22 and 23 may be a single or a double bond; Ris C-Calkyl, C-Ccycloalkyl, or C-Calkenyl; Rand Rare, for example, independently of each other hydrogen, C-Calkyl, C-Ccycloalkyl, C-Calkenyl, C-Calkynyl, aryl or heteroaryl; and, where applicable, to E/Z isomers, mixtures of E/Z isomers, diastereomers and/or tautomers, in each case in free form or in salt form; pesticidal compositions in which the active ingredient has been selected from those compounds and their tautomers; and a method of controlling pests using those compositions are described. 

Growing community of inventors

Basel, Switzerland

Fiona Murphy Kessabi