Kureha Corporation

Emiko Obata

Taiji Miyake

Nobuyuki Araki

Toru Yamazaki

Eiyu Imai

Kazuhiko Sunagawa

Hisashi Kanno

Provided is an azole derivative superior in disease-controlling activity contained as an active ingredient in agricultural or horticultural chemical agents. The azole derivative according to the present invention is represented by the following General Formula (I): (in Formula (I), Rrepresents an unsubstituted or substituted C-C-alkyl group;Rrepresents a carbonyl group-containing functional group, wherein the carbon atom in the carbonyl group is bound to the carbon atom in the cyclopentane ring substituted with Rand to a hydrogen atom, a hydroxyl group, R, OR, or NRR;Rand Reach represent a C-C-alkyl group, a C-C-alkenyl group, or a C-C-alkynyl group;Y represents a halogen atom, a C-C-alkyl group, a C-C-haloalkyl group, a C-C-alkoxy group, a C-C-haloalkoxy group, a phenyl group, a cyano group, or a nitro group;m is 0 to 5; andA represents a nitrogen atom or a methine group).

Azole derivative, method for producing same, intermediate compound, and agricultural or horticultural chemical agent and industrial material protecting agent

In order to provide a compound which exhibits a high controlling effect against plant diseases and is able to reduce phytotoxicity, the present invention is a triazole derivative represented by General Formula (I), the azole derivative being a (&#x2212;)-enantiomer or (+)-enantiomer having an &#x2014;Rgroup, hydroxy group, and substituted or unsubstituted benzyl group bonded to a cyclopentane ring in cis-form.

Azole derivative and uses thereof

In order to produce an intermediate from which a cyclic alcohol compound can be stereoselectively obtained, a method for producing an oxetane compound according to the present invention includes the step of reacting, with a cyanide salt, a compound represented by Formula (I): wherein Ris selected from a hydrogen atom and an alkyl group optionally having a substituent; Xis selected from a halogen atom and &#x2014;OSORwhere Ris selected from an alkyl group optionally having a substituent, a phenyl group, and a naphthyl group; and a ring Z1 represents a cyclic hydrocarbon optionally having a substituent, 

Method for manufacturing oxetane compound, method for manufacturing azolylmethylcyclopentanol compound, and intermediate compound

In order to provide a novel azole derivative, an azole derivative of the present invention is an azole derivative represented by a general formula (V'). (where Rand Rindependently represent a hydrogen atom, a C-Calkyl group, a phenyl group, or a benzyl group; X represents a halogen atom, a C-Calkyl group, a haloalkyl group, an alkoxy group or a haloalkoxy group, a phenyl group, a cyano group, or a nitro group; m represents an integer of 0 to 5; and A represents a nitrogen atom or a methyne group.)

Azole derivative, method for producing azole derivative, and intermediate compound

Provided is an azole derivative superior in disease-controlling activity contained as an active ingredient in agricultural or horticultural chemical agents. The azole derivative according to the present invention is represented by the following General Formula (I): 

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Tokyo, Japan

Emiko Obata