Smithkline Beecham Corporation

Glaxo Group Limited

Other

David Thomas Davies

Neil David Pearson

Graham Elgin Jones

Roger Edward Markwell

Ian Thomson Forbes

Laramie Mary Gaster

Paul Adrian Wyman

Keith Raymond Mulholland

William Henry Miller

Alan Joseph Hennessy

David Malcolm Duckworth

Andrew Lightfoot

Israil Pendrak

Robert A Daines

Timothy Francis Gallagher

Andrew Kenneth Takle

Jeffrey Michael Axten

Steven Dabbs

Timothy James Miles

Gerald Brooks

Francis D King

Mervyn Thompson

William Edward Bondinell

Roderick Alan Porter

Ilaria Giordano

Julia Castro Pichel

Joseph W Venslavsky

Peter Ham

Jose Maria Fiandor Roman

James A Chan

James B Hoffman

Angela Moghe

Laurence R Petrie

David Evan Davies

David Barros

Lihua Zhang

Nathalie Cailleau

Modesto J Remuiñan Blanco

Jason Anthony Rossi

Lihua(lily) Zhang

Lluis Ballell

Joel Michael Esken

Senthil Kumar Kusalakumari Sukumar

Modesto J Remuinan Blanco

Tricyclic nitrogen containing compounds and their use as antibacterials. Zand Zare independently selected from CH and N. 

Tricyclic nitrogen containing compounds as antibacterial agents

Bicyclic nitrogen containing compounds and their use as antibacterials.

Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones

Tricyclic nitrogen containing compounds of formula (I) and their use as antibacterials.

Heterocyclic compounds, their preparation and their use as antibacterials

Cyclohexane and cyclohexene derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly man.

Antibacterial compounds

Aminopiperidine derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man 

Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity

Piperidine derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man. The piperidine derivatives include compounds of formula (I): wherein R, AB, n, R, Rand Rare defined herein. For example, Ris an optionally substituted bicyclic carbocyclic or heterocyclic ring system, and Ris a group U-Rin which Ris an optionally substituted bicyclic heterocyclic ring system as defined herein (e.g. optionally substituted pyrido [3,2, -b][1,4] thiazin-yl).

Compounds

Piperidine derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man. 

Quinolines and nitrogenated derivative thereof substituted in 4-position by a piperidine-containing moiety and their use as antibacterial agents

Nitrogen-containing bicyclic heterocycles for use as antibacterials

Aminopiperidine derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man.

Aminopiperidine derivatives as antibacterials

Aminopiperidine quinolines and their azaisosteric analogues with antibacterical activity

The present invention relates to a compound of formula (I) or a pharmaceutically acceptable salt and/or N-oxide thereof:corresponding novel medicaments, pharmaceutical compositions and/or methods of

Quinoline derivatives as antibacterials

The invention relates to heterocyclic compounds having pharmacological activity, processes for their preparation, to compositions containing them and to their use in the treatment of CNS disorders such as anxiety.

Indole derivatives as 5-HT receptor antagonist

Piperidine derivatives and pharmaceutical derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man.

Quinoline derivatives and their use as antibacterial agents

A method of treating a CCR5-mediated disease state in mammals which comprises administering to a mammal in need of such treatment, an effective amount of a compound of formula (I) or a pharmaceutically acceptable salt thereof.

Compounds and methods

A compound of formula (I) or a salt thereof:

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Harlow, United Kingdom

David Thomas Davies