A. Nattermann & Cie Gmbh

Rhone-poulenc Rorer S.a.

Nattermann & Cie Gmbh

Armin Wendel

Miklos Ghyczy

Manfred Durr

Sigurd Leyck

Jorg Hager

Paul-Robert Imberge

Ulrich Posanski

Hans Betzing

Jurgen Biedermann

Jorg-Christian Hager

Helmut Wetzig

Volker Neuser

Kurt-Heinz Bauer

Volker Schulz

Jörg Hager

This invention relates to a pharmaceutical composition comprising as active principle, docetaxel or a taxoid derived from docetaxel, one or more unsaturated phospholipids and a small amount of one or more negative phospholipids, allow the active principle to be formulated in high concentration and are suitable for administration by injection.

Pharmaceutical composition based on taxoids

Pharmaceutical preparation containing phospholipids for the therapeutic treatment of rheumatic diseases which contain in addition to the antiphlogistically acting oxicam derivatives of the general formula ##STR1## special 1,2-diacyl-glycero-3-phosphocholines wherein 75-86% by weight of the acyl radicals are unsaturated fatty acid radicals, and the preparation thereof.

Pharmaceutical preparation for the therapeutic treatment of rheumatic

Pharmaceutical formulations for the treatment of gastrointestinal disorders, which contain as the active component an effective gastrointestinal disorder alleviating amount of a 1,2-diacylglycero-3-phosphocholine in which 75-86% by weight of the acyl radicals are unsaturated fatty acid radicals having a chain length of 16, 18 or 20 carbon atoms. The mixtures of fatty acid radicals in the acyl groups in the 1- and 2-positions preferably have different compositions. The formulations can also contain other active compounds, in particular those which display injurious gastrointestinal side effects.

Formulation with special 1,2-diacylglycero-3-phosphocholines for the

Phospholipid concentrates from natural or synthetic phospholipids and physiologically acceptable organic solvents and further additives of the following composition:

Phospholipid compositions and their use in plant protection spray

Liquid, active substance formulations containing an active substance insoluble or poorly soluble in water, or a mixture, a phospholipid, a special co-emulsifier (glycerinester in which the 1 or 2 OH groups have been esterized with hydrocarbon atoms of 8-16, preferably 8-10, C atoms by means of fatty acids and the 3 or remaining OH group of the glycerin body has been etherized with polyethyleneglycol, specifically, with 6-30, preferably 6-15 ethyleneoxide units) and a liquid carrier, the molar ratio of phospholipid to co-emulsifier being from 1:1 to 1:4, and the formulations being such that when added to water they form a transparent liquid system in the form of a microemulsion, with a degree of fineness of 10-200 nm in the lipid phase.

Liquid active ingredient concentrates for preparation of microemulsions

Process for the application of plant protectant spray mixtures in which the phospholipid concentrates are applied to open ground, phospholipids being discharged along with commercially available, diluted effective ingredient concentrates and the spray mixtures being formed before discharge from the active ingredient concentrate, water, and the phospholipid concentrate. This process employs packing units which contain the active ingredient concentrate and the appropriate quantity of phospholipid concentrate in separate compartments.

Process for the spray application of plant protective spray mixtures and

The invention provides N-propionylsarcosineanilides of the formula: ##STR1## wherein n is an integer of 1 to about 3 and the substituent A which can be the same or different when n is greater than 1 is selected from the group consisting of trifluoromethyl; halogen; nitro; acetyl; a straight-chain or branched alkyl group having 1 to 4 carbon atoms; a straight-chain or branched alkoxy group having 1 to 4 carbon atoms; a straight-chain or branched alkylmercapto group having 1 to 7 carbon atoms; a substituted alkylmercapto group of the formula: ##STR2## wherein n is an integer of 1 or 2, R.sub.1 can represent hydrogen and methyl, and R.sub.2 can represent hydroxyl, and an amino group of the formula:

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Cologne, Germany

Armin Wendel