Basf Aktiengesellschaft

Basf Se Corporation

Andreas Gypser

Thomas Grote

Siegfried Strathmann

Wassilios Grammenos

Eberhard Ammermann

Gisela Lorenz

Markus Gewehr

Hubert Sauter

Joachim Rheinheimer

Jordi Tormo I Blasco

Frank Schieweck

Reinhard Stierl

Bernd W M&uuml;ller

Peter Schäfer

Bernd Müller

Arne Ptock

Herbert Bayer

Ingo Rose

Volker Harries

Anja Schwögler

Roland G&ouml;tz

Oliver Cullmann

Franz R&ouml;hl

Carsten Blettner

Reinhard Kirstgen

Norbert G&ouml;tz

Ulrich Schöfl

Michael Rack

Peter Sch&auml;fer

Maria Scherer

Oliver Wagner

Norbert Götz

Siegried Strathmann

Oliver Cullman

Klaus J&uuml;ergen Pees

Rheinhard Stierl

Michael Keil

John-Bryan Speakman

Gerhard Hamprecht

Karl Eicken

Bernd Wolf

Klaus Oberdorf

Klaus Ditrich

Henry Van Tuyl Cotter

Horst Mayer

Keith Douglas Barnes

William Wakefield Wood

Yulin Hu

Thorsten Volk

Ruth M&uuml;ller

Adrian Steinmetz

Roland Götz

Gregory J Haley

Paul Carter

Franz Röhl

Günter Krummel

Jan Rether

Kathryn C Ferguson

J&uuml;rgen Curtze

Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula I in which

Substituted 6-(2-halogennphenyl)-triazolopyrimidines

5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings:

5-phenylpyrimidines, their preparation, intermediates for their preparation, and their use for controlling harmful fungi

The invention relates to 5-alkyl-7-aminotriazolopyrimidines of the formula (I) and to the salts thereof. In said formula substituents have the following meanings: Rand Reach is a hydrogen atom or a group of alkyl, alcenyl, haloalkyl, cycloalky, phenyl or naphtyle, saturated, unstaturated or aromatic heterocycle having from five to six members which contain from one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or Rand Rcan from together with a connecting them nitrogen atom a cycle of 5 to 6 members containing from one to four nitrogen atoms or from one to three nitrogen atoms and one sulfur or oxygen atom, Ris a cycloalkyl or bicycloalkyl group, R, Rand Rcan be substituted in conformity with a description, and X is an alkyl or alkyl halide group. The inventive methods and intermediary products necessary for producing said compounds, agents containing them and the use therefore for fighting against harmful mushroom are also disclosed. 

5-alkyl-7-aminotriazolopyrimidines, methods and intermediary product necessary for the production thereof, agents containing said compounds and the use thereof for fighting against harmful mushrooms

The invention relates to novel biphenyl carboxamides of formula (I), wherein A, R, Z, X, Y, m and n have the meanings given in the description, to multiple methods for producing these substances, to their use for combating unwanted micro-organisms and to novel intermediate products and the production thereof.

Trifluoromethyl-thiophene carboxylic acid aniledes and use thereof as fungicides

2-Substituted pyrimidines of the formula I in which the index n and the substituents L, R, R, R, R, R, R, A', A&#x2033; and A&#x2032;&#x2033; are as defined in the description and:

2-substituted pyrimidines

5-Phenylpyrimidines, their preparation, compositions comprising them and their use 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below:

5-Phenypyrimidines their preparation compositions comprising them and their use

5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below:

5-phenylpyrimidines, their preparation, compositions comprising them and their use

The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents Rto Rand L are as defined in the description and 

The invention relates to 2-(2-pyridyl)-5-phenyl-6-aminopyrimidines of formula I, wherein the substitutes and the index have the following meaning: Rrepresents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino. dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m=0 or 1-4; Rrepresents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R, Rrepresents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, Rand Rtogether with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; Rrepresents halogen, alkyl or halogenalkyl; Rrepresents hydrogen or one of the known groups in R; R, Rrepresent hydrogen, halogen, alkyl or halogenalkyl; Rrepresents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants 

2-(2-pyridyl)-5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi

The invention relates to 2-substituted pyrimidines of the formula I in which the index n and these substituents R, Rand Rare as defined in the description and Ris as defined below: where

2-Substituted pyrimidines

The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R, Rrepresent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or Rand Rcan, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; Rrepresents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby Rand Rcan be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by R. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.

7-amino triazolopyrimidines for controlling harmful fungi

Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n=0 or a whole number of 1-5; R=halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R=alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or Rbeing able to be substituted according to the description; R=alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi 

Fungicidal triazolopyrimidines, method for the production thereof and use thereof in controlling noxious fungi and agents containing said compounds

Z-substituted acrylamides of formula (I), where the substituents have the following meanings: X&#x2550;H, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, with X in the 3- or 4-position, n=1 or 2, where X can be different if n=2, R=alkyl, haloalkyl, cycloalkyl, alkoxy, haloalkoxy, aziridine and oxirane and R&#x2550;H, alkyl, haloalkyl, allyl, propargyl or CHC&#x2261;C-alkyl. Methods for production thereof, agents comprising the above and the use thereof for the treatment of plant-pathogenic fungal pests. 

Z-substituted acrylamides, methods for production thereof and agents comprising the same

The invention relates to 5-phenylpyrimidine of formula (I) wherein the substituents have the following designations: Rrepresents a five to ten-membered saturated, partially unsaturated or aromatic monocyclic or bicyclic heterocycle which contains between one and four heteroatoms from the group O, N or S, and which can be substituted as defined in the description; Rrepresents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; Rand Rrepresent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl; together with the nitrogen atom to which they are bonded, Rand Rcan also form a five or six-membered ring which can be split by a heteroatom and can carry at least one substituent; Rand Rrepresent hydrogen, halogen, alkyl, halogenalkyl or alkoxy; Rand Rrepresent hydrogen, halogen, alkyl or halogenalkyl; and Rrepresents hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, halogenalkoxy or alkoxycarbonyl. The invention also relates to methods and intermediate products for producing said compounds and the use of the same for controlling pathogenic fungi 

5-Phenylpyrimidines, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi

The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: Lrepresents cyano, S(&#x2550;O)Aor C(&#x2550;O)A, wherein Astands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; Astands for C&#x2013;Calkoxy, C&#x2013;Chaloalkoxy or one of the groups named in A; and n stands for 0, 1 or 2; L, Lrepresent hydrogen or halogen; L, Lrepresent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; Rrepresents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; Rrepresents hydrogen or R; Rand Rcan form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby Rand/or Rcan be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi. 

Fungicidal triazolopyrimidines, methods for producing the same, use thereof for combating harmful fungi and agents containing said substances

Growing community of inventors

Mannheim, Germany

Andreas Gypser